第六届中美华人有机化学教授会议（杭州，6月14-17日） 2010-06-12.pdf 
第六届中美华人有机化学教授会议（杭州，6月14-17日） 2010-06-12.pdf
Program The 6th Sino-US Chemistry Professors Conference: Organic Chemistry & Chemical Biology June 14 14,, 2010 (Monday) Time Program & Venue Location 8:00-18:00 Registration Santai Shan Hotel Lobby (三台山宾馆 大厅) jun Ren Hong Hongjun Yingxia Yuan 18:30-20:00 Welcome Reception Santai Shan Hotel: Bai-He Hall/百合厅, 1st Floor Prof. Yanguang Wang and Prof. Qian Wang 任红军：15868183766 Chairperson Section I: Organic Chemistry Location: Santai Shan, Tian-Liang Hall Hall//三台山，天朗厅,, 1st Floor June 15 15,, 2010 (Tuesday) Chairperson: Prof. Yanguang Wang (8:00-9:50) 8:30-8:50 Jeffrey Johnson (University of North Carolina at Chapel Hill) Complexity-Building Reactions: Recent Case Studies Weiping Tang (University of Wisconsin, Madison) 8:50-9:10 Stereoselective Addition of Halogen and Nucleophile to Unsaturated CarbonCarbon Bonds Aiwen Lei Lei（雷爱文,, 武汉大学） 9:10-9:30 Oxidative Coupling --- The Chemistry between Two Nucleophiles Hao Li (李浩，中科院上海药物研究所) 9:30-9:50 Gold(I) Catalyzed Dihydroamination of Allenes with Ureas Jie Wu (吴劼,, 复旦大学)) 9:50-10:15 基于 2-炔基苯甲醛的若干串联反应 Take Pictures and Coffee Break 8:00-8:30 Chairperson: Prof. Weiping Tang (10:15-11:55) 10:35-10:55 Gang Zhao (赵刚， 中科院上海有机化学研究所) 基于氨基酸的有机催化剂的设计、合成及其应用 Cheng Ma (马成， Zhejiang University) 10:55-11:15 Efficient Construction of Functionalized Spiro-3,4-dihydropyran Derivatives Xiaodong Shi (Department of Chemistry, West Virginia University) 11:15-11:35 1,2,3-Triazole, A Special Ligand in Tuning Transition Metal Catalyst Reactivity Wei Wang (University of New Mexico, Albuquerque, USA) 11:35-11:55 New Strategies in Developing Powerful Enantioselective Organocatalytic Cascade Jing Wu (吴静，杭州师范大学/Hangzhou Normal University) 10:15-10:35 A Highly Efficient Copper-Catalyzed Hydrosilylation System for the Asymmetric Synthesis of Valuable Chiral Alcohols 12:00-14:00 Lunch (Location: Santai Shan Hotel, Bai-He Hall/三台山，百合厅, 1st Floor)) Chairperson: Prof. Xiaodong Shi (14:00-15:50) 14:00-14:30 14:30-14:50 Zhangjie Shi (施章杰,, 北京大学） Recent Advances on C-O Activation Xigeng Zhou (周锡庚，复旦大学化学系) 14:50-15:10 Selective Insertions of C−H and N−H bonds of Organolanthanides and Their Application in Organic Synthesis Nan Zheng (University of Arkansas, Dept. of Chem. and Biochem.) Fe(II)-Catalyzed Intramolecular Amination of Aromatic C-H Bonds: Synthesis of 2,3-Disubstituted Indoles 15:10-15:30 15:30-15:50 Shuli You (游书力,, 中科院上海有机化学研究所) Ir-Catalyzed Allylic Substitution Reactions Huanfeng Jiang (江焕峰, South China University of Technology) 钯 催 化 炔 烃 溴 炔 化 反 应 研 究 /Palladium-Catalyzed Bromoalkynylation of Alkynes 15:50-16:05 Coffee Break Chairperson: Prof. Gang Zhao (16:05-17:45) 16:25-16:45 Chanjuan Xi (席婵娟, 清华大学) Multifaceted Reactivity of Organozirconates Lei Wang (王磊，淮北师范大学) 16:45-17:05 Cu(OTf)2-Catalyzed Arylmethylation of Terminal Alkynes with Benzylic Alcohols under Acid-, Base-, Ligand-, and Additive-Free Reaction Conditions Ning Jiao (焦宁,, 北京大学药学院天然药物及仿生药物国家重点实验室) 17:05-17:25 The Application of Dioxygen in Transition Metal Catalyzed Reactions Xingang Zhang (中科院上海有机化学研究所) 16:05-16:25 Pd-Catalyzed Direct Olefination and Benzylation of Highly Electron-Deficient Perfluoroarenes 17:25-17:45 Weiliang Duan Duan（段伟良,, 中科院上海有机化学研究所 ） Palladium-Catalyzed Asymmetric Addition of Diarylphosphines to Enones toward the Synthesis of Chiral Phosphines 18:00 Dinner (Location: Santai Shan Hotel, Bai-He Hall/三台山，百合厅, 1st Floor))) 17:00- Expo (Location: Santai Shan, Hai-Tang Hall Hall/三台山，海棠厅, Ground Floor) 19:30-- Scientific Advisory Board for Sino-US Chem Meeting (Location: Tea House at Santai Shan Lobby) Section II: Chemical Biology Location: Santai Shan, Hai-Tang Hall Hall//三台山，海棠厅,, Ground Floo Floorr June 15 15,, 2010 (Tuesday) Prof. Qian Wang (8:00-9:50) Chairperson：Prof. 8:30-8:50 Jianghong Rao (Stanford Medical School) A Biocompatible Condensation Reaction and Its Applications for Bioimaging Aimin Liu (Georgia State University) 8:50-9:10 Mechanistic Enzymology of Tryptophan Metabolism Pengfei Wang (University of Alabama at Birmingham) 9:10-9:30 Development of Glycosylation Method for Rapid Carbohydrate Synthesis Binghe Wang (Georgia State University) 8:00-8:30 9:30-9:50 9:50-10:15 Inhibitors of Hypoxia Inducible Factor-1α Yingfu Li (McMaster University, Canada) Engineering and Applications of DNAzymes Take Pictures and Coffee Break Chairperson: Prof. Zhanting Li (10:15-11:55) 10:35-10:55 Zhongwu Guo (Wayne State University) Chemoenzymatic Synthesis of GPI-Anchored Proteins and Glycoproteins Xuefei Huang (Michigan State University, Department of Chemistry) 10:55-11:15 Magnetic Glyco-nanoparticles: Applications in Detections of Cancer and Atherosclerosis Ning-Hua Tan (Kunming Institute of Botany, CAS) 11:15-11:35 Discovery and Mechanism of Antitumor Cyclopeptides from Rubia Yunnanensis Ching-Hwa Kiang （Rice University, Houston, TX, USA） 11:35-11:55 Probing Protein and DNA Interaction Forces Using Single-Molecule Nanobiology Ao Zhang Zhang(张翱,, 中科院上海药物研究所) 10:15-10:35 Natural Products-Inspired Drug Design & Discovery 12:00-14:00 Lunch (Location: Santai Shan,, Bai-He Hall/三台山，百合厅, 1st Floor)) Chairperson: Prof. Jianghong Rao (14:00-15:50) 14:30-14:50 Steven Benner (The Foundation for Applied Molecular Evolution and The Westheimer Institute for Science and Technology） Synthesizing Artificial Genetic Systems Chuan He (The University of Chicago) 14:50-15:10 DNA/RNA Oxidative Modification by the Human AlkB Type Proteins Zhen Huang (Department of Chemistry, Georgia State University, Atlanta, 14:00-14:30 Georgia 30303, USA) Probing High Fidelity of DNA Base Paring via Selenium Atomic Probe and 3D Crystal Structure 15:10-15:30 15:30-15:50 Huaqiang Zeng (National University of Singapore) Circularly Folded Aromatic Pentamers and Their Biological Implications Zhongjun Li (李中军,, 北京大学药学院) Studies on the Methodology of the Quickly Assembly of High-mannose Oligosaccharides Based on the Hydrophobically Assisted Switching-Phase (HASP) Strategy 15:50-16:05 Coffee Break 16:25-16:45 Chairperson: Prof. Zhen Xi (16:05-17:45) Qian Wang (University of South Carolina)) Viral assemblies as substrates for cell culturing Guigen Li (Texas Tech University) 16:45-17:05 Asymmetric Catalytic Strecker Reaction of N-Phosphonyl Imines Using NonToxic Cyanide Sources and BINOL-Derived Catalysts Xi Chen (Department of Chemistry, University of California-Davis) 17:05-17:25 Efficient Chemoenzymatic Synthesis of Complex Carbohydrates Chengzhi Cai (University of Houston) 16:05-16:25 Biofunctionalization of Silicon and Biomaterials 17:25-17:45 Xuelong Sun (孙学龙，Cleveland State University) Spherical Glycosurface Assembling Based Intact Immobilized Liposome 18:00 Dinner (Santai Shan, Bai-He Hall/三台山，百合厅, 1st Floor) 17:00-- Expo (Location: Santai Shan, Hai-Tang Hall Hall/三台山，海棠厅, Ground Floor) 19:30-- Scientific Advisory Board for Sino-US Chem Meeting (Location: Tea House at Santai Shan Lobby) Section I: Organic Chemis try Chemistry Location: Santai Shan, Tian-Liang Hall Hall//三台山，天朗厅,, 1st Floor June 16 16,, 2010 (Wednesday Wednesday)) Chairperson: Prof. Biao Yu (8:00-9:50) 8:30-8:50 Yong Qing (秦勇,, 四川大学) Total Synthesis and SAR Study of Anti-MRSA Marinopyrrole A Richard P. Hsung (University of Wisconsin-Madison) 8:50-9:10 Total Synthesis of Phomactin A Wei-Min Dai (Zhejiang University & The Hong Kong University of Science and 9:10-9:30 Technology) Total Synthesis via Ring-Closing Metathesis Approaches Yongmin Liang (梁永民,, 兰州大学) 8:00-8:30 Electrophile-Induced Tandem Cyclization Reactions for the Annulation of Heterocycles 9:30-9:50 贾彦兴 (北京大学药学院、天然药物及仿生药物国家重点实验室) Total Synthesis of (-)-Stephanotic Acid Methyl Ester and (-)-Celogentin C 9:50-10:10 Coffee Break Chairperson: Prof. Richard P. Hsung (10:10-11:50) 10:30-10:50 Biao Yu (俞飚， 中科院上海有机化学研究所) 环状三萜皂甙的高效合成及其抗肿瘤活性 Biao Jiang (姜标，Shanghai Institute of Organic Chemistry, CAS) 10:50-11:10 Study on the Synthesis of Palauamine and Its Derivatives Bo Liu (刘波，四川大学化学学院) 11:10-11:30 Total Synthesis of Heliespirones A & C Song Yang (杨松, 贵州大学精细化工研究开发中心/Guizhou University) 11:30-11:50 Synthesis and Bioactivity of Heterocyclic Thioether, Sulfoxide, and Sulfone Derivatives Xiaoguang Lei (雷晓光,, 北京生命科学研究所/天津大学) 10:10-10:30 Exploring the Structural Diversity and Biological Activity of Complex Natural Products 12:00-14:00 Lunch (Location: Santai Shan, Bai-He Hall/三台山，百合厅, 1st Floor) Chairperson: Prof. Wei Wang (14:00-15:50) 14:00-14:30 14:30-14:50 Kuiling Ding (丁奎岭, 中科院上海有机研究所） Highly Efficient Chiral Organometallic Catalysts for Homo- and Heterogeneous Asymmetric Hydrogenation Chunjiang Wang (王春江, 武汉大学化学与分子科学学院) Organocatalyzed Asymmetric Michael Addition of α-Aryl Ketone to Nitroolefins for Construction of Adjacent Quaternary and Tertiary Stereocenters 14:50-15:10 15:10-15:30 Song Ye (叶松, 中科院化学所/Institute of Chemistry, CAS) Asymmetric Cycloaddition Reactions of Ketenes Catalyzed by N-Heterocyclic Carbenes Zhaoguo Zhang (张兆国, 上海交通大学化学化工学院) The Design and Application of Chiral Ligands in Asymmetric Hydrogenation Reactions 15:30-15:50 Junan Ma (马军安, 天津大学化学系) Application of Novel Chiral Phase-Transfer Catalysts in Asymmetric Synthesis 15:50-16:05 Coffee Break Chairperson: Prof. Rui Wang (16:05-17:45) 16:25-16:45 Baoan Song (宋宝安, Guizhou University) Enantioselective Synthesis and Antiviral Activity of Novel β-Amino Esters by Mannich Reaction Minghua Xu (徐明华，中国科学院上海药物研究所 ) 16:45-17:05 Access to Enantioenriched Homoallylamines Nucleophilic Allylation of N-Sulfinyl Imines Guan-Wu Wang (王官武, 中国科学技术大学) 16:05-16:25 by Efficient Asymmetric Solvent-Free Reactions Promoted by Ball Milling 17:25-17:45 Yingchun Chen (陈应春,, 四川大学华西药学院) Asymmetric Allylic Alkylation Promoted by Lewis Basic Organocatalysts Wanbing Zhang ( 张 万 斌 ， School of Chemistry and Chemical Engineering, 18:00 Shanghai Jiao Tong University) Development of Effective Axial Chiral Ligands and Catalysis with New Design Concept for Asymmetric Catalysis Location: Liu-Tong Hotel, Tian-Fu Ju Banquet (Location: Ju//六通宾馆，天府居,, 1st Floor Floor) 17:05-17:25 Section II: Organic Chemistry & Chemical Biology Location: Hai-Tang Hall Hall//海棠厅,, Ground Floor June 16 16,, 2010 (Wednesday Wednesday)) Chairperson: Prof. Jinbo Hu (8:00-9:50) 8:00-8:30 Sukbok Chang (Korea Advanced Institute of Science and Technology)) Metal-Mediated C-H Bond Activation of Heterocycles for the C-C and C-N Bond Formation 8:30-8:50 Liming Zhang （University of California, Santa Barbara） Gold-Catalyzed Efficient Formation of Saturated N-Heterocycles 8:50-9:10 Kung K. Wang (Department of Chemistry, West Virginia University, Morgantown) Synthesis of a Basket-Shaped C56H38 Hydrocarbon as a Precursor Toward and End-Cap Template for Carbon [6, 6]Nanotube Lei Liu (刘磊，Tsinghua University) 9:10-9:30 New methods for chemical synthesis of proteins Guosheng Liu (刘国生, Shanghai Institute of Organic Chemistry) 9:30-9:50 Palladium-Catalyzed Aminofluorination of Alkenes 9:50-10:10 Coffee Break 10:10-11:50 Chairperson: Prof. Liming Zhang （10:10-11:50 10:10-11:50） 10:30-10:50 Fengling Qing (卿凤翎,, 中国科学院上海有机化学研究所) Fluoroalkylation of C-H bonds Ruimao Hua (华瑞茂,, 清华大学化学系) 10:50-11:10 原子经济性环化加成反应设计与研究 Shujiang Tu (屠树江,, 徐州师范大学) 11:10-11:30 多组分反应的化学选择性研究 Zhixiang Xie (谢志翔,, 兰州大学化学化工学院) 11:30-11:50 Total Synthesis of Biyouyanagin A Zhi-Zhen Huang ( 黄 志 真 ， School of Chemistry and Chemical Engineering, 10:10-10:30 Nanjing University) Cascade Reactions by the Combinations of Transition Metal and Organocatalysis 12:00-14:00 Lunch (Location: Santai Shan, Bai-He Hall/三台山，百合厅, 1st Floor)) Chairperson: Prof. Baoan Song (14:00-15:50) 14:30-14:50 Hongbin Zhang Zhang（张洪彬，云南大学） 一些生物活性分子的设计与合成研究 Hao Fang (School of Pharmacy, Shandong University) 14:50-15:10 Pyrrolidine-based drug discovery Chen Hongyu (Nanyang Technological University) 14:00-14:30 15:10-15:30 Fabrication of Complex Nanostructures by Colloidal Chemistry Yaxiong Tang (唐亚雄,, 中国科学院成都生物研究所) Anti-Cancer Potential of Flavokawains on Human Cancer 15:30-15:50 15:50-16:05 Xuechen Li (Department of Chemistry, The University of Hong Kong) Development of New Methodology in the Chemical Synthesis (Glyco)peptides/(glyco)proteins of Coffee Break Chairperson: Prof. Zhangjie Shi (16:05-17:45) 16:25-16:45 Zhen Xi (席真，南开大学元素有机化学研究所) Ribosome Translocation and Antibiotics Xiaoqin Zhu (朱晓晴,, 南开大学化学学院) 16:45-17:05 Thermodynamic Diagnoses of Properties and Mechanism of Imines as Hydride Acceptors in Acetonitirle with “Molecule ID Card” Biwu Ma (The Molecular Foundry, Lawrence Berkeley National Laboratory) 16:05-16:25 Organic Solar Cells with Solution Processable Materials 17:25-17:45 Zhishu Huang (黄志纾, 中山大学药学院) Turning off Transcription of the Bcl-2 Gene by Stabilizing the Bcl-2 Promoter Quadruplex with Quindoline Derivatives Zhuo Tang (唐卓,, 中科院成都生物所) 18:00 In Vitro Selection of DNA-Cleaving DNA Enzyme Which Could Work at Physiological Condition Location: Liu-Tong Hotel, Tian-Fu Ju Banquet (Location: Ju//六通宾馆，天府居,, 1st Floor Floor) 17:05-17:25 Section I: Organic Chemistry Location: Santai Shan, Tian-Liang Hall Hall//三台山，天朗厅,, 1st Floor June 17 17,, 2010 (Thursday) Chairperson: Prof. Hongbin Zai (8:00-9:50) 8:00-8:30 8:30-8:50 Zhanting Li (黎占亭,, 中国科学院上海有机化学研究所) Exploring the Applications of Proorganized Oligomers and Polymers in Developing Functional Materials Yuanjiang Pan (潘远江，Zhejiang University) 电喷雾质谱中离子/中性复合物中间体介导的新型电荷转移反应研究 9:10-9:30 Ruikang Tang (唐睿康，Zhejiang University)) Carboxyl-mediated crystallization of calcium minerals in a biomimetic system Yong Ju (巨勇,, 清华大学化学系) 9:30:9-50 新型含甾体/三萜骨架功能分子的合成与性能研究 Yan Zhang (张艳,, 南京大学化学化工学院) 9:50-10:05 Smart Self-Assembling System Based on Modified Short Peptides Coffee Break 8:50-9:10 Chairperson: Prof. Feihe Huang (10:05-11:35) 10:35-10:55 Jinbo Hu Hu（胡金波,, 中国科学院上海有机化学研究所） New Fluoroolefination Reactions Based on Fluorinated Sulfone and Sulfoximine Reagents Zhiqiang Wang （Kent State University） 10:55-11:15 Catalytic Activities of Bacterial Nitric Oxide Synthase Baoqing Song (宋庆宝,, 浙江工业大学化材学院) 10:05-10:35 Asymmetric Henry Reaction Catalyzed by Cu(I)-based Chiral Amino Alcohol Complex 11:15-11:35 12:00-13:00 Xinjing Tang (汤新景,, 北京大学医学部天然药物及仿生药物国家重点实验室) Photomodulating RNA Cleavage Using Photolabile Circular Antisense Oligodeoxynucleotides Lunch (Location: Santai Shan, Bai-He Hall/三台山，百合厅, 1st Floor)) Section II: Supramolecular and Material Chemistry Location: Santai Shan, Hai-Tang Hall Hall//三台山，海棠厅,, Ground Floo Floorr June 17 17,, 2010 (Thursday) Chairperson: Prof. Guanwu Wang (8:00-9:50) 8:30-8:50 Yi Liu (Lawrence Berkeley National Laboratory) Donors and Acceptors Made to Order – from Interlocked Molecules to Supramolecular Materials Feihe Huang (Zhejiang University) 8:50-9:10 Threaded Structures Based on Crown Ether Derivatives Jingsong You (游劲松,, 四川大学化学学院) 9:10-9:30 Discovery of Fluorescent Core Skeletons Based on Heteroaromatics and their application in Supramolecular Chemistry Jun Li (National University of Singapore) 9:30-9:50 Supramolecular Self-Assembled Macromolecular Systems for Biomaterials Application Hua Zhang (Nanyang Technological University) 9:50-10:05 Nanopatterns and Nanomaterials: Fabrication, Synthesis and Applications Chemistry Coffee Break 8:00-8:30 Yuanjiang Pan (10:15-11:45) Chairperson: Prof. Prof.Yuanjiang 10:25-10:45 Chuan-Feng Chen (陈传峰,, 中国科学院化学研究所) Hydrogen Bonds Mediated Self-Assembly Based on Hydrazide Derivatives Dunwei Wang (Boston College, Department of Chemistry) 10:45-11:05 Energy Interconversion Using Nanomaterials: Challenges and Opportunities Derong Cao ( 曹 德 榕 , School of Chemistry and Chemical Engineering, South 11:05-11:25 China University of Technology) Synthesis and Electroluminescence Properties of Diketopyrrolopyrrole-Containing Polymers Qichun Zhang (MSE, Nanyang Technological University) 11:25-11:45 Organic Materials for OLED Leyong Wang (王乐勇,, 南京大学化学化工学院) 10:05-10:25 分子陀螺的合成与组装 12:00-13:00 Lunch (Location: Santai Shan,, Bai-He Hall/三台山，百合厅, 1st Floor))